Repare Therapeutics Inc. Patent Applications Pending
22 applications still open at the USPTO, newest filing first, as the USPTO Open Data Portal records them; the company is the first-named applicant. The application number opens the full record at Patent Center.
- 2025-09-26: Application 19469929; Invention METHODS OF DETERMINING GENOMIC COPY NUMBER ALTERATIONS; Applicant REPARE THERAPEUTICS INC.; Status Docketed New Case - Ready for Examination.
- 2025-06-16: Application 19139501; Invention METHODS OF MAKING 2-AMINO-1-(3-HYDROXY-2,6-DIMETHYLPHENYL)-5,6-DIMETHYL-1H-PYRROLO-[2,3-B]PYRIDINE-3-CARBOXAMIDE, A MYT1 INHIBITOR; Applicant Repare Therapeutics Inc.; Status Application Undergoing Preexam Processing.
- 2025-02-12: Application 19051391; Invention COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING COMPOUNDS AND OF THEIR USE AS ATR KINASE INHIBITORS; Applicant Repare Therapeutics Inc.; Status Docketed New Case - Ready for Examination.
- 2024-11-18: Application 18866842; Invention HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME; Applicant Repare Therapeutics Inc.; Status Non Final Action Mailed.
| Filed | Application | Invention | Applicant | Status | Published as | Inventor name | Inventor country | Examiner |
|---|---|---|---|---|---|---|---|---|
| 2025-09-26 | 19469929 | METHODS OF DETERMINING GENOMIC COPY NUMBER ALTERATIONS | REPARE THERAPEUTICS INC. | Docketed New Case - Ready for Examination | US20260250751A1 | Elia Aguado-Fraile Adam Petrone Jorge Reis-Filho Victoria Rimkunas Artur Veloso | Canada Canada Canada Canada Canada | CENTRAL, DOCKET |
| 2025-06-16 | 19139501 | METHODS OF MAKING 2-AMINO-1-(3-HYDROXY-2,6-DIMETHYLPHENYL)-5,6-DIMETHYL-1H-PYRROLO-[2,3-B]PYRIDINE-3-CARBOXAMIDE, A MYT1 INHIBITOR | Repare Therapeutics Inc. | Application Undergoing Preexam Processing | Angelos DOVLETOGLOU Robert Charles LIVINGSTON Jill A. CAPUTO Sarah M. POUND Qi GAO | United States United States United States United States United States | ||
| 2025-02-12 | 19051391 | COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING COMPOUNDS AND OF THEIR USE AS ATR KINASE INHIBITORS | Repare Therapeutics Inc. | Docketed New Case - Ready for Examination | US20250179070A1 | Sheldon N. CRANE Vouy Linh Truong Abbas Abdoli Jean-François Truchon Cameron Black Stéphane Dorich Lee Fader Stéphanie Lanoix Paul Jones Miguel St-Onge Audrey Picard Cyrus M. Lacbay | Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada | CENTRAL, DOCKET |
| 2024-11-18 | 18866842 | HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME | Repare Therapeutics Inc. | Non Final Action Mailed | US20250304537A1 | Cameron BLACK Janek SZYCHOWSKI Bingcan LIU Evelyne DIETRICH Frédéric VALLÉE Simon SURPRENANT Alexander PERRYMAN Sheldon N. CRANE Vouy Linh TRUONG Alexanne BOUCHARD Abbas ABDOLI Frederic IZQUIERDO Dominique BELLA NDONG Stephane CIBLAT Francis BARABE Thomas PINTER | Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada | RICCI, CRAIG D |
| 2024-10-04 | 18854217 | METHODS OF USING ATR INHIBITORS | Repare Therapeutics Inc. | Non Final Action Mailed | US20250228862A1 | Theo GOULLET DE RUGY Stephen MORRIS Jordan YOUNG Michal ZIMMERMANN Dominik GLODZIK | Canada Canada Canada Canada United States | PECKHAM, RICHARD GRANT |
| 2024-08-22 | 18840582 | POLO-LIKE KINASE 4 (PLK4) INHIBITORS, PHARMACEUTICAL COMPOSITIONS, METHODS OF PREPARATION AND USES THEREOF | Repare Therapeutics Inc. | Non Final Action Mailed | US20250177396A1 | Frédéric VALLÉE Boubacar SOW Monica BUBENIK Michel GALLANT Philippe MOCHIRIAN Simon SURPRENANT Martin DUPLESSIS Bingcan LIU Alexander PERRYMAN | Canada Canada Canada Canada Canada Canada Canada Canada Canada | CLARK, AMY LYNN |
| 2023-12-14 | 18540119 | USE OF ATR INHIBITORS IN COMBINATION WITH PARP INHIBITORS FOR TREATING CANCER | Repare Therapeutics Inc. | Non Final Action Mailed | US20240173330A1 | Cameron Black Michal Zimmermann | Canada Canada | ENGLISH, CONNOR KENNEDY |
| 2023-10-25 | 18288308 | METHODS OF TREATING CANCERS HAVING A BIALLELIC LOSS OF FUNCTION OR GENE OVEREXPRESSION MUTATION | Repare Therapeutics Inc. | Non Final Action Mailed | US20240392379A1 | Jorge Sergio REIS Maria KOEHLER Victoria RIMKUNAS Dominik GLODZIK Michael ZINDA Robert DABER Ian SILVERMAN | United States United States United States United States United States United States United States | BAUSCH, SARAE L |
| 2023-10-02 | 63541936 | COMBINATION THERAPIES INCLUDING MYT1 INHIBITORS AND WEE1 INHIBITORS | Repare Therapeutics Inc. | Provisional Application Expired | David GALLO Michal ZIMMERMANN Stephen MORRIS Jimmy FOURTOUNIS Gary MARSHALL | Canada Canada Canada Canada United States | ||
| 2023-10-02 | 63541935 | MYT1 INHIBITORS FOR THE TREATMENT OF CANCERS HARBORING REPLICATION STRESS MUTATIONS | Repare Therapeutics Inc. | Provisional Application Expired | Artur VELOSO Jimmy FOURTOUNIS Gary MARSHALL | United States Canada United States | ||
| 2023-09-18 | 63583510 | COMBINATION TREATMENT OF CANCERS | REPARE THERAPEUTICS INC. | Provisional Application Expired | Michal Zimmermann Anne Roulston Julia Yang Danielle Ulanet | Canada Canada United States United States | ||
| 2023-03-28 | 63455221 | METHODS OF DETERMINING GENOMIC COPY NUMBER ALTERATIONS | Repare Therapeutics Inc. | Provisional Application Expired | Elia AGUADO-FRAILE Adam PETRONE Jorge REIS-FILHO Victoria RIMKUNAS Artur VELOSO | United States United States United States United States United States | ||
| 2022-10-03 | 17916760 | COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING COMPOUNDS AND OF THEIR USE | Repare Therapeutics Inc. | Docketed New Case - Ready for Examination | US20230151014A1 | Janek SZYCHOWSKI Bingcan LIU Evelyne DIETRICH Frédéric VALLÉE Alexander PERRYMAN Jean-François TRUCHON Robert PAPP Patrick BEAULIEU | Canada Canada Canada Canada Canada Canada Canada Canada | FERGUSON, JALISA HOLMES |
| 2022-04-29 | 63336827 | QUINAZOLINONES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME | Repare Therapeutics Inc. | Provisional Application Expired | Janek SZYCHOWSKI Bingcan LIU Evelyne DIETRICH Alexander PERRYMAN Sheldon N. CRANE Vouy-linh TRUONG Abbas ABDOLI Alexanne BOUCHARD | Canada Canada Canada Canada Canada Canada Canada Canada | ||
| 2021-10-06 | 63253004 | TRICYCLIC HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME | Repare Therapeutics Inc. | Provisional Application Expired | Janek SZYCHOWSKI Evelyne DIETRICH Frédéric VALLÉE | Canada Canada Canada | ||
| 2021-10-06 | 63252961 | COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING COMPOUNDS AND OF THEIR USE | Repare Therapeutics Inc. | Provisional Application Expired | Janek SZYCHOWSKI Bingcan LIU Evelyne DIETRICH Frédéric VALLÉE Alexander PERRYMAN Jean-François TRUCHON Robert PAPP Patrick BEAULIEU Vouy-Linh TRUONG Kaveh MATINKHOO Sheldon N. CRANE | Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada | ||
| 2021-10-04 | 63251942 | COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING COMPOUNDS AND OF THEIR USE | Repare Therapeutics Inc. | Provisional Application Expired | Janek SZYCHOWSKI Bingcan LIU Evelyne DIETRICH Frédéric VALLÉE Alexander PERRYMAN Jean-François TRUCHON Robert PAPP Patrick BEAULIEU Vouy-Linh TRUONG Kaveh MATINKHOO Sheldon N. CRANE | Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada Canada | ||
| 2020-12-11 | PCTUS2020064662 | USE OF ATR INHIBITORS IN COMBINATION WITH PARP INHIBITORS | REPARE THERAPEUTICS INC. | PCT - International Search Report Mailed to IB | MICHAL ZIMMERMANN MARIA KOEHLER ANNE ROULSTON | Canada United States Canada | THOMAS, SHANE M | |
| 2019-12-11 | 62946876 | USE OF ATR INHIBITORS IN COMBINATION WITH PARP INHIBITORS | Repare Therapeutics Inc. | Provisional Application Expired | Michal ZIMMERMANN Anne ROULSTON Maria KOEHLER | Canada Canada United States | ||
| 19613726 | CRYSTALLINE FORMS, CRYSTALLINE SALT FORMS, COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME | Repare Therapeutics Inc. | Application Undergoing Preexam Processing | Angelos Dovletoglou Robert Charles Livingston Song Xue Dansu Li Kimberly Miller | United States United States United States United States Canada | |||
| 19525148 | COMBINATION THERAPIES INCLUDING MYT1 INHIBITORS AND WEE1 INHIBITORS | Repare Therapeutics Inc. | Application Undergoing Preexam Processing | David Gallo Michal Zimmermann Stephen Morris Jimmy Fourtounis Gary Marshall | Canada Canada Canada Canada United States | |||
| 19525144 | MYT1 INHIBITORS FOR THE TREATMENT OF CANCERS HARBORING REPLICATION STRESS MUTATIONS | REPARE THERAPEUTICS INC. | Application Undergoing Preexam Processing | Artur Veloso Jimmy Fourtounis Gary Marshall | United States Canada United States |