G1 THERAPEUTICS, INC. Active Patents
51 granted patents the USPTO still lists as patented, newest filing first, as the USPTO Open Data Portal records them; the company is the first-named applicant. The application number opens the full record at Patent Center.
- 2022-05-11: Application 17742315; Invention SUBSTITUTED 1',2'-DIHYDRO-3'H-SPIRO[CYCLOHEXANE-1,4'-PYRIMIDO[5',4':4,5]PYRROLO[2,1-c][1,2,4]TRIAZIN]-3'-ONES AS CYCLIN-DEPENDENT KINASE INHIBITORS; Applicant G1 Therapeutics, Inc.; Status Patented Case.
- 2022-02-28: Application 17683146; Invention MORPHIC FORMS OF G1T38 AND METHODS OF MANUFACTURE THEREOF; Applicant G1 Therapeutics, Inc.; Status Patented Case.
- 2021-04-21: Application 17236687; Invention MORPHIC FORMS OF TRILACICLIB AND METHODS OF MANUFACTURE THEREOF; Applicant G1 Therapeutics, Inc.; Status Patented Case.
- 2021-04-05: Application 17222873; Invention TRANSIENT PROTECTION OF NORMAL CELLS DURING CHEMOTHERAPY; Applicant G1 Therapeutics, Inc.; Status Patented Case.
| Filed | Application | Invention | Applicant | Status | Granted | Patent | Published as | Inventor name | Inventor country | Examiner |
|---|---|---|---|---|---|---|---|---|---|---|
| 2022-05-11 | 17742315 | SUBSTITUTED 1',2'-DIHYDRO-3'H-SPIRO[CYCLOHEXANE-1,4'-PYRIMIDO[5',4':4,5]PYRROLO[2,1-c][1,2,4]TRIAZIN]-3'-ONES AS CYCLIN-DEPENDENT KINASE INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2023-05-09 | 11643416 | US20220306644A1 | Jay Copeland Strum | United States | WILLIS, DOUGLAS M |
| 2022-02-28 | 17683146 | MORPHIC FORMS OF G1T38 AND METHODS OF MANUFACTURE THEREOF | G1 Therapeutics, Inc. | Patented Case | 2024-11-12 | 12139494 | US20230043305A1 | Alexander Smith Hannah S. White Patricia Andres Xufeng Sun Lei Zhu Petinka I. Vlahova | United States United States United States United States United States United States | MCDOWELL, BRIAN E |
| 2021-04-21 | 17236687 | MORPHIC FORMS OF TRILACICLIB AND METHODS OF MANUFACTURE THEREOF | G1 Therapeutics, Inc. | Patented Case | 2024-12-17 | 12168666 | US20210387993A1 | Stephen Schneider Alexander Smith Hannah S. White Jay Copeland Strum Jaroslaw Mazurek | United States United States United States United States Netherlands | DAHLIN, HEATHER RAQUEL |
| 2021-04-05 | 17222873 | TRANSIENT PROTECTION OF NORMAL CELLS DURING CHEMOTHERAPY | G1 Therapeutics, Inc. | Patented Case | 2023-08-08 | 11717523 | US20210299130A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2021-02-24 | 17184354 | SYNTHESIS OF 1,4-DIAZASPIRO[5.5]UNDECAN-3-ONE | G1 Therapeutics, Inc. | Patented Case | 2023-07-25 | 11708337 | US20210179567A1 | Stephen E. Schneider Hannah White Thomas Fessard Sagar Beldar | United States United States Switzerland Switzerland | RAO, DEEPAK R |
| 2021-02-22 | 17181638 | HSPC-SPARING TREATMENTS FOR RB-POSITIVE ABNORMAL CELLULAR PROLIFERATION | G1 Therapeutics, Inc. | Patented Case | 2023-05-23 | 11654148 | US20210213022A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis X. Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2020-12-14 | 17121392 | SYNTHESIS OF N-(HETEROARYL)-PYRROLO[3,2-D]PYRIMIDIN-2-AMINES | G1 Therapeutics, Inc. | Patented Case | 2023-04-18 | 11629150 | US20210122755A1 | Alexander Smith Hannah S. White Francis Xavier Tavares Sergiy Krasutsky Jian-Xie Chen Roberta L. Dorrow Hua Zhong | United States United States United States United States United States United States United States | YOO, SUN JAE |
| 2020-11-13 | 17097854 | MORPHIC FORMS OF TRILACICLIB AND METHODS OF MANUFACTURE THEREOF | G1 Therapeutics, Inc. | Patented Case | 2021-04-27 | 10988479 | Stephen Schneider Alexander Smith Hannah S. White Jay Copeland Strum Jaroslaw Mazurek | United States United States United States United States Netherlands | ZHANG, YANZHI | |
| 2020-07-08 | 16924033 | G1T38 SUPERIOR DOSAGE REGIMES | G1 Therapeutics, Inc. | Patented Case | 2022-06-14 | 11357779 | US20200405721A1 | Andrew Beelen Jay Copeland Strum | United States United States | LEESER, ERICH A |
| 2020-05-28 | 16886309 | TRANSIENT PROTECTION OF NORMAL CELLS DURING CHEMOTHERAPY | G1 Therapeutics, Inc. | Patented Case | 2021-06-22 | 11040042 | US20200345742A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2020-05-13 | 15931330 | CDK INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2021-02-23 | 10927120 | US20200277300A1 | Francis X. Tavares Jay Copeland Strum | United States United States | MURRAY, JEFFREY H |
| 2019-12-19 | 16721631 | MORPHIC FORMS OF G1T38 AND METHODS OF MANUFACTURE THEREOF | G1 Therapeutics, Inc. | Patented Case | 2022-03-01 | 11261193 | US20200123168A1 | Alexander Smith Hannah S. White Patricia Andres Xufeng Sun Lei Zhu Petinka I. Vlahova | United States United States United States United States United States United States | MCDOWELL, BRIAN E |
| 2019-09-16 | 16572418 | TREATMENT OF RB-NEGATIVE TUMORS USING TOPOISOMERASE INHIBITORS IN COMBINATION WITH CYCLIN DEPENDENT KINASE 4/ | G1 Therapeutics, Inc. | Patented Case | 2021-08-17 | 11090306 | US20200022983A1 | Jay Copeland Strum John E. Bisi Patrick Joseph Roberts Jessica A. Sorrentino | United States United States United States United States | SCHMITT, MICHAEL J |
| 2019-06-05 | 16432244 | PRESERVATION OF IMMUNE RESPONSE DURING CHEMOTHERAPY REGIMENS | G1 Therapeutics, Inc. | Patented Case | 2022-12-20 | 11529352 | US20190321370A1 | Jessica A. Sorrentino Anne Y. Lai Jay C. Strum Patrick Joseph Roberts | United States United States United States United States | PUTTLITZ, KARL J |
| 2019-01-22 | 16254364 | ANTI-NEOPLASTIC COMBINATIONS AND DOSING REGIMENS USING CDK4/ | G1 Therapeutics, Inc. | Patented Case | 2022-09-20 | 11446295 | US20190151311A1 | Jay Copeland Strum John E. Bisi Patrick Joseph Roberts Jessica A. Sorrentino Hannah S. White | United States United States United States United States United States | RAMACHANDRAN, UMAMAHESWARI |
| 2018-12-21 | 16230412 | PYRIMIDINE-BASED COMPOUNDS FOR THE TREATMENT OF CANCER | G1 Therapeutics, Inc. | Patented Case | 2020-04-14 | 10618905 | US20190119294A1 | Jay Copeland Strum | United States | PAGANO, ALEXANDER R |
| 2018-12-21 | 16230396 | SUBSTITUTED DIHYDROPYRAZINO[1',2':1,5]PYRROLO[2,3-d]PYRIMIDINE-BASED ANTIPROLIFERATIVE AGENTS | G1 Therapeutics, Inc. | Patented Case | 2020-11-10 | 10829490 | US20190135811A1 | Jay Copeland Strum David Jung | United States United States | WILLIS, DOUGLAS M |
| 2018-12-21 | 16230388 | ANTIPROLIFERATIVE PYRIMIDINE-BASED COMPOUNDS | G1 Therapeutics, Inc. | Patented Case | 2020-05-19 | 10654831 | US20190135784A1 | Jay Copeland Strum Ricky D. Gaston Robert C. Gadwood | United States United States United States | SACKEY, EBENEZER O |
| 2018-12-21 | 16230381 | SYNTHESIS OF N-(HETEROARYL)-PYRROLO[3,2-D]PYRIMIDIN-2-AMINES | G1 Therapeutics, Inc. | Patented Case | 2020-12-15 | 10865210 | US20190135820A1 | Alexander Smith Hannah S. White francis Xavier Tavares Sergiy Krasutsky Jian-Xie Chen Roberta L. Dorrow Hua Zhong | United States United States United States United States United States United States United States | YOO, SUN JAE |
| 2018-12-20 | 16228308 | Highly Active Anti-Neoplastic and Anti-Proliferative Agents | G1 Therapeutics, Inc. | Patented Case | 2020-07-14 | 10709711 | US20190125752A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | JEAN-LOUIS, SAMIRA JM |
| 2018-12-19 | 16226430 | CDK INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2020-06-30 | 10696682 | US20190119292A1 | Francis X. Tavares Jay Copeland Strum | United States United States | MURRAY, JEFFREY H |
| 2018-11-01 | 16178419 | HSPC-SPARING TREATMENTS FOR RB-POSITIVE ABNORMAL CELLULAR PROLIFERATION | G1 Therapeutics, Inc. | Patented Case | 2021-02-23 | 10925878 | US20190070185A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2018-09-26 | 16142574 | TREATMENT OF RB-NEGATIVE TUMORS USING TOPOISOMERASE INHIBITORS IN COMBINATION WITH CYCLIN DEPENDENT KINASE 4/ | G1 Therapeutics, Inc. | Patented Case | 2019-09-17 | 10413547 | US20190030034A1 | Jay Copeland Strum John E. Bisi Patrick Joseph Roberts Jessica A. Sorrentino | United States United States United States United States | CHU, YONG LIANG |
| 2018-08-24 | 16112362 | HSPC-SPARING TREATMENTS FOR RB-POSITIVE ABNORMAL CELLULAR PROLIFERATION | G1 Therapeutics, Inc. | Patented Case | 2019-10-08 | 10434104 | US20180360841A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2018-08-24 | 16112360 | TRANSIENT PROTECTION OF NORMAL CELLS DURING CHEMOTHERAPY | G1 Therapeutics, Inc. | Patented Case | 2021-04-06 | 10966984 | US20180360840A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2018-04-02 | 15943278 | TRANSIENT PROTECTION OF NORMAL CELLS DURING CHEMOTHERAPY | G1 Therapeutics, Inc. | Patented Case | 2020-05-26 | 10660896 | US20180221378A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis X. Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2018-03-12 | 15918877 | CDK INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2019-01-29 | 10189851 | US20180201619A1 | Francis X. Tavares Jay C. Strum | United States United States | MURRAY, JEFFREY H |
| 2018-03-12 | 15918852 | CDK INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2019-01-29 | 10189850 | US20180201618A1 | Francis X. Tavares Jay C. Strum | United States United States | MURRAY, JEFFREY H |
| 2018-03-12 | 15918834 | CDK Inhibitors | G1 Therapeutics, Inc. | Patented Case | 2019-01-29 | 10189849 | US20180201617A1 | Francis X. Tavares Jay C. Strum | United States United States | MURRAY, JEFFREY H |
| 2018-01-02 | 15860483 | LACTAM KINASE INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2019-11-05 | 10464940 | US20180127431A1 | Francis Xavier Tavares | United States | PATEL, SAGAR S |
| 2017-07-31 | 15665071 | TRICYCLIC LACTAMS FOR USE IN HSPC-SPARING TREATMENTS FOR RB-POSITIVE ABNORMAL CELLULAR PROLIFERATION | G1 Therapeutics, Inc. | Patented Case | 2019-08-13 | 10376519 | US20170333440A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Ricky D. Gaston Robert C. Gadwood | United States United States United States United States United States | JEAN-LOUIS, SAMIRA JM |
| 2017-03-13 | 15457699 | ANTI-NEOPLASTIC COMBINATIONS AND DOSING REGIMENS USING CDK4/ | G1 Therapeutics, Inc. | Patented Case | 2019-03-19 | 10231969 | US20170182043A1 | Jay Copeland Strum John E. Bisi Patrick Joseph Roberts Jessica A. Sorrentino Hannah S. White | United States United States United States United States United States | KATAKAM, SUDHAKAR |
| 2016-12-21 | 15387083 | HSPC-Sparing Treatments for RB-Positive Abnormal Cellular Proliferation | G1 Therapeutics, Inc. | Patented Case | 2018-09-18 | 10076523 | US20170100405A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2016-11-10 | 15348862 | LACTAM KINASE INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2018-01-02 | 9856268 | US20170057972A1 | Francis Xavier Tavares | United States | PATEL, SAGAR S |
| 2016-11-10 | 15348770 | CDK Inhibitors | G1 THERAPEUTICS, INC. | Patented Case | 2018-05-01 | 9957276 | US20170057971A1 | Francis X. Tavares Jay C. Strum | United States United States | MURRAY, JEFFREY H |
| 2016-11-03 | 15342990 | Transient Protection of Normal Cells During Chemotherapy | G1 THERAPEUTICS, INC. | Patented Case | 2018-10-02 | 10085992 | US20170065597A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2016-10-07 | 15288878 | TRANSIENT PROTECTION OF NORMAL CELLS DURING CHEMOTHERAPY | G1 Therapeutics, Inc. | Patented Case | 2018-04-03 | 9931345 | US20170037051A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2015-12-29 | 14982443 | Lactam Kinase Inhibitors | G1 Therapeutics, Inc. | Patented Case | 2017-08-29 | 9745316 | US20160108054A1 | Francis Xavier Tavares | United States | PATEL, SAGAR S |
| 2015-05-14 | 14712630 | CDK Inhibitors | G1 Therapeutics, Inc. | Patented Case | 2016-11-01 | 9481691 | US20150246926A1 | Francis X. Tavares Jay C. Strum | United States United States | MURRAY, JEFFREY H |
| 2015-05-14 | 14712582 | CDK Inhibitors | G1 Therapeutics, Inc. | Patented Case | 2016-11-22 | 9499564 | US20150246925A1 | Francis X. Tavares Jay C. Strum | United States United States | MURRAY, JEFFREY H |
| 2015-04-17 | 14690180 | Tricyclic Lactams for Use in HSPC-Sparing Treatments for RB-Positive Abnormal Cellular Proliferation | G1 THERAPEUTICS, INC. | Patented Case | 2017-08-01 | 9717735 | US20150299212A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Ricky D. Gaston Robert C. Gadwood | United States United States United States United States United States | JEAN-LOUIS, SAMIRA JM |
| 2014-09-26 | 14498796 | LACTAM KINASE INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2016-02-16 | 9260442 | US20150018348A1 | Francis Xavier Tavares | United States | PATEL, SAGAR S |
| 2014-08-05 | 14452296 | CDK Inhibitors | G1 Therapeutics, Inc. | Patented Case | 2015-08-11 | 9102682 | US20150031880A1 | Francis X. Tavares Jay C. Strum | United States United States | MASHA, OLUWAFEMI L |
| 2014-03-14 | 14214048 | HSPC-Sparing Treatments for RB-Positive Abnormal Cellular Proliferation | G1 THERAPEUTICS, INC. | Patented Case | 2016-12-27 | 9527857 | US20140271466A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2014-03-14 | 14212911 | Transient Protection of Normal Cells During Chemotherapy | G1 Therapeutics, Inc. | Patented Case | 2016-10-11 | 9464092 | US20140275067A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2014-03-14 | 14212430 | Transient Protection of Normal Cells During Chemotherapy | G1 Therapeutics, Inc. | Patented Case | 2016-11-08 | 9487530 | US20140275066A1 | Jay Copeland Strum John Emerson Bisi Patrick Joseph Roberts Francis Xavier Tavares | United States United States United States United States | TRAN, MY CHAU T |
| 2014-01-23 | 14162649 | CDK INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2014-09-02 | 8822683 | US20140142299A1 | Francis X. Tavares Jay C. Strum | United States United States | MASHA, OLUWAFEMI L |
| 2014-01-23 | 14162637 | CDK INHIBITORS | G1 Therapeutics, Inc. | Patented Case | 2014-09-09 | 8829012 | US20140142306A1 | Francis X. Tavares Jay C. Strum | United States United States | MASHA, OLUWAFEMI L |
| 2013-04-24 | 13869594 | CDK INHIBITORS | G1 THERAPEUTICS, INC. | Patented Case | 2014-04-08 | 8691830 | US20130237534A1 | Francis X. Tavares Jay C. Strum | United States United States | MASHA, OLUWAFEMI L |
| 2013-04-24 | 13869576 | CDK INHIBITORS | G1 THERAPEUTICS, INC. | Patented Case | 2013-12-03 | 8598197 | US20130237533A1 | Francis X. Tavares Jay C. Strum | United States United States | MASHA, OLUWAFEMI L |
| 2013-04-24 | 13869520 | CDK INHIBITORS | G1 THERAPEUTICS, INC. | Patented Case | 2013-12-03 | 8598186 | US20130237544A1 | Francis X. Tavares Jay C. Strum | United States United States | MASHA, OLUWAFEMI L |