Advertisement
Screener

LIGAND PHARMACEUTICALS INCORPORATED (LGND) Patents: Active

LIGAND PHARMACEUTICALS INCORPORATED Active Patents

93 granted patents the USPTO still lists as patented, newest filing first, as the USPTO Open Data Portal records them; the company is the first-named applicant. The application number opens the full record at Patent Center.

  • 2024-03-05: Application 18595919; Invention USE OF THYROID BETA-AGONISTS; Applicant Metabasis Therapeutics, Inc.; Status Patented Case.
  • 2023-06-23: Application 18340177; Invention TOPICAL ANTIVIRAL COMPOSITIONS, DELIVERY SYSTEMS, AND METHODS OF USING THE SAME; Applicant Ligand Pharmaceuticals Incorporated; Status Patented Case.
  • 2023-03-22: Application 18246284; Invention ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME; Applicant CYDEX PHARMACEUTICALS, INC.; Status Patented Case.
  • 2022-10-19: Application 17996613; Invention BENZYLOXY PHOSPH(ON)ATE COMPOUNDS; Applicant Ligand Pharmaceuticals Incorporated; Status Patented Case.
FiledApplicationInventionApplicantStatusGrantedPatentPublished asInventor nameInventor countryExaminer
2024-03-0518595919USE OF THYROID BETA-AGONISTSMetabasis Therapeutics, Inc.
Viking Therapeutics, Inc.
Patented Case2025-10-1412440502US20250000880A1
Brian Lian
Rochelle Hanley
Misha DINERMAN
Mark Erion
Serge Boyer
Hongjian Jiang
United States
United States
United States
United States
United States
China
RAMACHANDRAN, UMAMAHESWARI
2023-06-2318340177TOPICAL ANTIVIRAL COMPOSITIONS, DELIVERY SYSTEMS, AND METHODS OF USING THE SAMELigand Pharmaceuticals IncorporatedPatented Case2025-09-0212403087US20230330008A1
Kimberly McHale
Ryan Doxey
Nathan Stasko
United States
United States
United States
MAEWALL, SNIGDHA
2023-03-2218246284ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAMECYDEX PHARMACEUTICALS, INC.Patented Case2026-08-0412698348US20230357451A1
Vincent D. ANTLE
Andre FERNANDES
Mariana RODRIGUES
Claudio VILELA
United States
Portugal
Portugal
Portugal
WARD, PAUL V
2022-10-1917996613BENZYLOXY PHOSPH(ON)ATE COMPOUNDSLigand Pharmaceuticals IncorporatedPatented Case2026-02-1712552820US20230159574A1
Lin Zhi
United States
MCINTOSH III, TRAVISS C
2022-06-0817835828NUCLEOTIDE PRODRUG COMPOUNDSLigand Pharmaceuticals IncorporatedPatented Case2023-01-3111566041US20220298198A1
Lin Zhi
United States
BERRY, LAYLA D
2022-05-1117776199ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAMECyDex Pharmaceuticals, Inc.Patented Case2026-07-0712674005US20230002513A1
Vincent D. Antle
United States
CRAIGO, BAHAR ALAWI
2022-05-0617738621USE OF THYROID BETA-AGONISTSMetabasis Therapeutics, Inc.
Viking Therapeutics, Inc.
Patented Case2024-04-0911951114US20220257618A1
BRIAN LIAN
Rochelle Hanley
Misha Dinerman
Mark Erion
Serge Boyer
Hongjian Jiang
United States
United States
United States
United States
United States
China
RAMACHANDRAN, UMAMAHESWARI
2021-10-2817513093HETEROCYCLE AMINES AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2023-10-0311773110US20220119413A1
Koc-Kan Ho
David Diller
Jeffrey J. Letourneau
Brian F. McGuinness
Andrew G. Cole
David Rosen
Cornelis A. van Oeveren
Jason C. Pickens
Lin Zhi
Yixing Shen
Bijan Pedram
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
KIFLE, BRUCK
2021-10-1817604729CRYSTALLINE FORMS AND METHODS OF PRODUCING CRYSTALLINE FORMS OF A COMPOUNDLigand Pharmaceuticals IncorporatedPatented Case2025-06-0312319651US20220204448A1
Lin Zhi
Henri Sasmor
United States
United States
ISMAIL, REHANA
2021-09-0317465929TUNABLE NITRIC OXIDE-RELEASING MACROMOLECULES HAVING MULTIPLE NITRIC OXIDE DONOR STRUCTURESLigand Pharmaceuticals Incorporated
The University of North Carolina at Chapel Hill
Patented Case2025-12-2312503428US20210395191A1
Mark Schoenfisch
Yuan Lu
Nathan Stasko
Jian Bao
United States
United States
United States
United States
XU, JIANGTIAN
2021-07-2817387929NASAL AND OPHTHALMIC DELIVERY OF AQUEOUS CORTICOSTEROID SOLUTIONSCyDex Pharmaceuticals, Inc.Patented Case2025-07-2912370352US20220339414A1
James D. Pipkin
Rupert O. Zimmerer JR.
John M. Siebert
United States
United States
United States
WERTZ, ASHLEE ELIZABETH
2021-01-1417148785Azetidine DerivativesLigand UK Development LimitedPatented Case2025-03-1112246014US20210267974A1
Stephen Roughley
Steven Walls
Terance Hart
Rachel Parsons
Paul Brough
Christopher Graham
Alba Macias
United Kingdom
United Kingdom
United Kingdom
United Kingdom
United Kingdom
United Kingdom
United Kingdom
COPPINS, JANET L
2020-11-2417103328FRACTIONATED ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAMECyDex Pharmaceuticals, Inc.Patented Case2023-10-2411795241US20210147582A1
Vincent D. Antle
Charles Alan Watson
David W. Miles
United States
United States
United States
MAIER, LEIGH C
2020-10-1517071273IMIDAZO-FUSED HETEROCYCLES AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2024-01-0211858938US20210040102A1
Lin Zhi
United States
KANTAMNENI, SHOBHA
2020-09-1517021909SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONSCyDex Pharmaceuticals, Inc.Patented Case2023-11-0711806402US20210093727A1
Vincent D. Antle
United States
OLSON, ANDREA STEFFEL
2020-08-1216969521GLUCAGON RECEPTOR ANTAGONISTSLIGAND PHARMACEUTICALS INCORPORATEDPatented Case2025-01-2812208071US20210121422A1
Lin Zhi
Ian Henderson
Joseph Kaloko
Martin Osterhout
United States
United States
United States
United States
COFFA, SERGIO
2020-08-0316983617SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2022-06-1411358931US20200361866A1
Lin Zhi
United States
MCDOWELL, BRIAN E
2020-07-1016925926METHODS AND COMPOSITIONS ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTORLigand Pharmaceuticals, Inc.Patented Case2022-08-1611413274US20210046045A1
Lin Zhi
Keith Marschke
Virginia H. Grant
Steven L. Roach
Yixing Shen
Jason C. Pickens
Bijan Pedram
Cornelis Arjan van Oeveren
Lino J. Valdez
Andrew R. Hudson
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
JACKSON, SHAWQUIA
2020-07-0816960681ACETAL COMPOUNDS AND THERAPEUTIC USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2024-04-3011970482US20200339551A1
Lin Zhi
United States
SEAMAN, D MARGARET M
2020-05-1516875855DPI FORMULATION CONTAINING SULFOALKYL ETHER CYCLODEXTRINCyDex Pharmaceuticals, Inc.Patented Case2022-10-1111464862US20200276314A1
James D. Pipkin
Gerold L. Mosher
Douglas B. Hecker
United States
United States
United States
HIRT, ERIN E
2020-01-2416752400MANUFACTURING PROCESS FOR CYCLODEXTRIN DERIVATIVESCyDex Pharmaceuticals, Inc.Patented Case2021-12-2811208500US20200157252A1
Vincent D. Antle
Jose R. Matos
United States
United States
OLSON, ANDREA STEFFEL
2020-01-0716735988HETEROCYCLE AMINES AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2021-11-3011186593US20200216468A1
Koc-Kan Ho
David Diller
Jeffrey J. Letourneau
Brian F. McGuinness
Andrew G. Cole
David Rosen
Cornelis A. van Oeveren
Jason C. Pickens
Lin Zhi
Yixing Shen
Bijan Pedram
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
KIFLE, BRUCK
2019-12-2716728840Injectable Nitrogen Mustard Compositions Comprising a Cyclodextrin Derivative and Methods of Making and Using the SameCydex Pharmaceuticals, Inc.Patented Case2020-12-1510864183US20200268698A1
James D. Pipkin
Stephen G. Machatha
United States
United States
ARNOLD, ERNST V
2019-11-0116672170COMPOSITION CONTAINING SULFOALKYL ETHER CYCLODEXTRIN AND LATANOPROSTCyDex Pharmaceuticals, Inc.Patented Case2022-09-0611433082US20200179400A1
Naomi Esaki
James D. Pipkin
United States
United States
BABSON, NICOLE PLOURDE
2019-09-1616572493METHODS AND COMPOSITIONS FOR MODULATING HORMONE LEVELSLigand Pharmaceuticals IncorporatedPatented Case2020-12-2910874638US20200009112A1
Lin Zhi
United States
WEDDINGTON, KEVIN E
2019-08-3016557768PRODRUG COMPOUNDS AND THEIR USESLIGAND PHARMACEUTICALS INCORPORATEDPatented Case2022-03-2211278559US20190388452A1
Lin Zhi
United States
LEWIS, PATRICK T
2019-03-1416333576FORMULATIONS CONTAINING ACETAMINOPHEN AND SULFOALKYL ETHER CYCLODEXTRINCyDex Pharmaceuticals, Inc.Patented Case2026-01-2012527755US20190255000A1
James D. Pipkin
Gerold L. Mosher
Roger A. Rajewski
United States
United States
United States
CHONG, YONG SOO
2019-02-2816289241GLUCAGON ANTAGONISTSMetabasis Therapeutics, Inc.Patented Case2022-06-0711352321US20190330144A1
Jorge E GOMEZ-GALENO
Scott J. HECKER
Qun DANG
Mali Venkat REDDY
Zhili SUN
Matthew P. GROTE
Thanh Huu NGUYEN
Robert Huerta LEMUS
Haiqing LI
United States
United States
United States
United States
United States
United States
United States
United States
United States
JAVANMARD, SAHAR
2019-02-0816271735SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS AND METHODS OF PREPARATION THEREOFCyDex Pharmaceuticals, Inc.Patented Case2020-07-0710703826US20190169316A1
James D. Pipkin
Gerold L. Mosher
Douglas B. Hecker
United States
United States
United States
OLSON, ANDREA STEFFEL
2018-12-0516210561INHALANT FORMULATION CONTAINING SULFOALKYL ETHER CYCLODEXTRIN AND CORTICOSTEROIDCyDex Pharmaceuticals, Inc.Patented Case2020-10-1310799599US20190105404A1
James D. PIPKIN
Rupert O. ZIMMERER
Diane O. THOMPSON
Gerold L. MOSHER
United States
United States
United States
United States
HAGHIGHATIAN, MINA
2018-11-1916195782THYROMIMETICS FOR THE TREATMENT OF FATTY LIVER DISEASESMetabasis Therapeutics, Inc.Patented Case2021-02-2310925885US20190083515A1
Edward E. Cable
Mark D. Erion
United States
United States
KATAKAM, SUDHAKAR
2018-11-0516181233SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONSCyDex Pharmaceuticals, Inc.Patented Case2020-09-2210780177US20190070303A1
Vincent D. Antle
United States
OLSON, ANDREA STEFFEL
2018-10-1916095228USE OF THYROID BETA-AGONISTSMetabasis Therapeutics, Inc.
Viking Therapeutics, Inc.
Patented Case2022-06-0711351183US20190321379A1
Brian Lian
Rochelle Hanley
Misha Dinerman
Mark Erion
Serge Boyer
Hongjian Jiang
United States
United States
United States
United States
United States
China
RAMACHANDRAN, UMAMAHESWARI
2018-10-0116148798SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2020-08-0410730831US20190040006A1
Lin Zhi
United States
MCDOWELL, BRIAN E
2018-09-1016126199METHODS AND COMPOSITIONS ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTORLigand Pharmaceuticals, Inc.Patented Case2020-08-1110736875US20180369197A1
Lin Zhi
Keith Marschke
Virginia H. Grant
Steven L. Roach
Yixing Shen
Jason C. Pickens
Bijan Pedram
Cornelis Arjan van Oeveren
Lino J. Valdez
Andrew R. Hudson
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
JACKSON, SHAWQUIA
2018-08-0816058778THYROID HORMONE RECEPTOR AGONIST AND USE THEREOFMetabasis Therapeutics, Inc.Patented Case2019-09-2410420781US20180344752A1
Mark Erion
Hongjian Jiang
Serge Henri Boyer
United States
China
United States
SHTERENGARTS, SAMANTHA L
2018-08-0216053550ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAMECyDex Pharmaceuticals, Inc.Patented Case2020-10-1310800861US20180346609A1
Vincent D. Antle
Álvaro Lopes
Daniel Monteiro
United States
Portugal
Portugal
OLSON, ANDREA STEFFEL
2018-07-2416043833FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USECydex Pharmaceuticals, Inc.Patented Case2019-12-2410512697US20180326090A1
Gerold L. Mosher
Rebecca L. Wedel
Karen T. Johnson
Stephen G. Machatha
Jane A. Cowee
Daniel J. Cushing
United States
United States
United States
United States
United States
United States
SHIAO, REI TSANG
2018-07-0216025199INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE 1 (DGAT-1) AND USES THEREOFMetabasis Therapeutics, Inc.Patented Case2020-07-1410709718US20180303856A1
K. Raja Reddy
Jeff Stebbins
Serge H. Boyer
Mark D. Erion
Scott J. Hecker
Nicholas Brian Raffaele
Brett C. Bookser
Venkat Reddy Mali
United States
United States
United States
United States
United States
United States
United States
United States
MURRAY, JEFFREY H
2018-06-2216015925HETEROCYCLE AMINES AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2020-03-3110604533US20180298031A1
Koc-Kan Ho
David Diller
Jeffrey J. Letourneau
Brian F. McGuinness
Andrew G. Cole
David Rosen
Cornelis A. van Oeveren
Jason C. Pickens
Lin Zhi
Yixing Shen
Bijan Pedram
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
KIFLE, BRUCK
2018-06-1116005601PRODRUG COMPOUNDS AND USES THEROFLigand Pharmaceuticals Inc.Patented Case2018-12-1110150788US20180291050A1
Lin Zhi
United States
ROZOF, TIMOTHY R
2018-02-2815908504METHODS OF TREATMENT ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTORLIGAND PHARMACEUTICALS INCORPORATEDPatented Case2019-09-2410420748US20180185333A1
Keith B. Marschke
Lin Zhi
United States
United States
WEDDINGTON, KEVIN E
2017-11-1715817056INHALANT FORMULATION CONTAINING SULFOALKYL ETHER CYCLODEXTRIN AND CORTICOSTEROIDCyDex Pharmaceuticals, Inc.Patented Case2019-02-1910207008US20180154015A1
James D. Pipkin
Rupert O. Zimmerer
Diane O. Thompson
Gerold L. Mosher
United States
United States
United States
United States
SCHLIENTZ, NATHAN W
2017-09-2915721556GLUCAGON ANTAGONISTSMetabasis Therapeutics, Inc.Patented Case2019-03-0510221130US20180022695A1
Jorge E. Gomez-Galeno
Scott J. Hecker
Qun Dang
Mali Venkat Reddy
Zhili Sun
Matthew P. Grote
Thanh Huu Nguyen
Robert Huerta Lemus
Haiqing Li
United States
United States
United States
United States
United States
United States
United States
United States
United States
MATOS NEGRON, TAINA DEL MAR
2017-08-3115693248MANUFACTURING PROCESS FOR CYCLODEXTRIN DERIVATIVESCyDex Pharmaceuticals, Inc.Patented Case2020-04-2810633462US20180051098A1
Vincent D. Antle
Jose R. Matos
United States
United States
OLSON, ANDREA STEFFEL
2017-08-2515687407METHOD FOR TREATING DISORDERS ASSOCIATED WITH GLOMERULAR FUNCTIONLigand Pharmaceuticals Inc.Patented Case2018-06-129993461US20170354646A1
Jinkun Zhang
Zofia E. Dziewanowska
Rene Belder
Ian Henderson
Joseph B. Bogardus
Zhaoying Zhang
United States
United States
United States
United States
United States
United States
HARTSFIELD, KATHRIEN ANN
2017-05-0915590884SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2018-10-2310106500US20170247325A1
Lin Zhi
United States
MCDOWELL, BRIAN E
2017-05-0915590813DERIVATIVES OF URIDINE 5'-CYCLOPHOSPHATE USEFUL TO TREAT HEPATITIS C VIRAL INFECTIONSLigand Pharmaceuticals IncorporatedPatented Case2018-06-1910000522US20170334942A1
Lin Zhi
United States
MCINTOSH III, TRAVISS C
2017-03-0915454967FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USECydex Pharmaceuticals, Inc.Patented Case2018-07-3110034947US20170173178A1
Gerold L. Mosher
Rebecca L. Wedel
Karen T. Johnson
Stephen G. Machatha
Jane A. Cowee
Daniel J. Cushing
United States
United States
United States
United States
United States
United States
SHIAO, REI TSANG
2017-03-0215448411SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS AND METHODS OF PREPARATION THEREOFCYDEX PHARMACEUTICALS, INC.Patented Case2019-02-1210202468US20170172926A1
James D. Pipkin
Gerold L. Mosher
Douglas B. Hecker
United States
United States
United States
OLSON, ANDREA STEFFEL
2017-02-2115505428FRACTIONATED ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAMECyDex Pharmaceuticals, Inc.Patented Case2020-12-0110851184US20170275388A1
Vincent D. Antle
Charles Alan Watson
David W. Miles
United States
United States
United States
MAIER, LEIGH C
2016-12-2915323080PRODRUG COMPOUNDS AND USES THEROFLIGAND PHARMACEUTICALS, INC.Patented Case2018-06-129994600US20170158725A1
Lin Zhi
United States
ROZOF, TIMOTHY R
2016-11-1415351272ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAMECydex Pharmaceuticals, Inc.Patented Case2019-06-1810323103US20170158781A1
Vincent D. Antle
Alvaro Lopes
Daniel Monteiro
United States
Portugal
Portugal
OLSON, ANDREA STEFFEL
2016-08-2515247164METHODS AND COMPOSITIONS ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTORLigand Pharmaceuticals, Inc.Patented Case2018-10-3010111859US20160374989A1
Lin Zhi
Keith Marschke
Virginia H. Grant
Steven L. Roach
Yixing Shen
Jason C. Pickens
Bijan Pedram
Cornelius Arjan van Oeveren
Lino J. Valdez
Andrew R. Hudson
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
JACKSON, SHAWQUIA
2016-08-1215118821PRODRUG COMPOUNDS AND THEIR USESLIGAND PHARMACEUTICALS, INC.Patented Case2019-10-2210449210US20170056429A1
Lin Zhi
United States
LEWIS, PATRICK T
2016-08-1015233748SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONSCyDex Pharmaceuticals, Inc.Patented Case2017-09-059750822US20160346405A1
Vincent D. Antle
United States
MAIER, LEIGH C
2016-07-1415111741METHODS AND COMPOSITIONS FOR MODULATING HORMONE LEVELSLIGAND PHARMACEUTICALS INCORPORATEDPatented Case2019-10-1510441567US20160338995A1
Lin Zhi
United States
WEDDINGTON, KEVIN E
2016-06-1315181190PHARMACEUTICAL COMPOSITIONS COMPRISING PRASUGREL AND CYCLODEXTRIN DERIVATIVES AND METHODS OF MAKING AND USING THE SAMECYDEX PHARMACEUTICALS, INC.Patented Case2018-10-3010111863US20170007586A1
Gerold L. Mosher
Stephen G. Machatha
Daniel J. Cushing
United States
United States
United States
MAIER, LEIGH C
2016-05-1115151740INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE 1 (DGAT-1) AND USES THEREOFMETABASIS THERAPEUTICS, INC.Patented Case2018-07-3110034891US20160263132A1
K. RAJA REDDY
JEFF STEBBINS
SERGE H. BOYER
MARK D. ERION
SCOTT J. HECKER
NICHOLAS BRIAN RAFFAELE
BRETT C. BOOKSER
VENKAT REDDY MALI
United States
United States
United States
United States
United States
United States
United States
United States
MURRAY, JEFFREY H
2016-05-0515034757DERIVATIVES OF URIDINE 5'-CYCLOPHOSPHATE USEFUL TO TREAT HEPATITIS C VIRAL INFECTIONSLIGAND PHARMACEUTICALS INCORPORATEDPatented Case2017-06-139676809US20160347783A1
Lin Zhi
United States
MCINTOSH III, TRAVISS C
2016-03-1515070718IMIDAZO-FUSED HETEROCYCLES AND USES THEREOFLigand Pharmaceuticals, Inc.Patented Case2020-10-2010807983US20160297824A1
Lin Zhi
United States
KANTAMNENI, SHOBHA
2016-01-2615006940HETEROCYCLE AMINES AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2018-07-2410030034US20160347767A1
Koc-Kan Ho
David Diller
Jeffrey J. Letourneau
Brian F. McGuinness
Andrew G. Cole
David Rosen
Cornelis A. van Oeveren
Jason C. Pickens
Lin Zhi
Yixing Shen
Bijan Pedram
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
KIFLE, BRUCK
2015-11-3014954772SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONSCyDex Pharmaceuticals, Inc.Patented Case2018-11-0610117951US20160158384A1
Vincent D. Antle
United States
OLSON, ANDREA STEFFEL
2015-09-1114775587METHODS OF TREATMENT ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTORLIGAND PHARMACEUTICALS INCORPORATEDPatented Case2018-05-089962370US20160022638A1
Keith B. Marschke
Lin Zhi
United States
United States
WEDDINGTON, KEVIN E
2015-09-0414846049FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USECydex Pharmaceuticals, Inc.Patented Case2017-04-189623045US20160058786A1
Gerold L. Mosher
Rebecca L. Wedel
Karen T. Johnson
Stephen G. Machatha
Jane A. Cowee
Daniel J. Cushing
United States
United States
United States
United States
United States
United States
SHIAO, REI TSANG
2015-08-1414827228SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2017-06-139675583US20160038461A1
Lin Zhi
United States
MCDOWELL, BRIAN E
2015-05-1514713930HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USESLIGAND PHARMACEUTICALS INC.Patented Case2017-04-189622991US20150252043A1
Lin Zhi
Andrew R. Hudson
Cornelis A. Van Oeveren
Steven L. Roach
Bijan Pedram
Yixing Shen
Lino J. Valdez
Jillian Basinger
Virginia Heather Sharron Grant
Jason C. Pickens
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
SHTERENGARTS, SAMANTHA L
2015-04-2114437439ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAMECYDEX PHARMACEUTICALS, INC.Patented Case2018-08-0710040872US20150284479A1
Vincent D. Antle
Álvaro Lopes
Daniel Monteiro
United States
Portugal
Portugal
OLSON, ANDREA STEFFEL
2015-03-1314428151NOVEL NUCLEOTIDE PRODRUG COMPOUNDS AND USELIGAND PHARMACEUTICALS INC.Patented Case2016-05-039326991US20150246068A1
Lin Zhi
K. Raja Reddy
United States
United States
MCINTOSH III, TRAVISS C
2015-02-2514631768METHOD FOR TREATING GLOMERULOSCLEROSISLigand Pharmaceuticals Inc.Patented Case2017-05-309662312US20150164865A1
Jinkun Zhang
Zofia E. Dziewanowska
Rene Belder
Ian Henderson
Joseph B. Bogardus
Zhaoying Zhang
United States
United States
United States
United States
United States
United States
HARTSFIELD, KATHRIEN ANN
2015-02-2314628373INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE 1 (DGAT-1) AND USES THEREOFMETABASIS THERAPEUTICS, INC.Patented Case2016-05-179340566US20150166590A1
K. RAJA REDDY
JEFF STEBBINS
SERGE H. BOYER
MARK D. ERION
SCOTT J. HECKER
NICHOLAS BRIAN RAFFAELE
BRETT C. BOOKSER
VENKAT REDDY MALI
United States
United States
United States
United States
United States
United States
United States
United States
MURRAY, JEFFREY H
2014-12-2914585073NOVEL ACTIVATORS OF GLUCOKINASEMetabasis Therapeutics, Inc.Patented Case2016-12-209522926US20150119365A1
Feng Tian
Qun Dang
G. Sridhar Prasad
Wenyu Li
Brett C. Bookser
Nicholas Brian Raffaele
Mark D. Erion
United States
United States
United States
United States
United States
United States
United States
BALASUBRAMANIAN, VENKATARAMAN
2014-11-2614555503GLUCAGON ANTAGONISTSMetabasis Therapeutics, Inc.Patented Case2017-10-109783494US20150087680A1
Jorge E. Gomez-Galeno
Scott J. Hecker
Qun Dang
Mali Venkat Reddy
Zhili Sun
Matthew P. Grote
Thanh Huu Nguyen
Robert Huerta Lemus
Haiqing Li
United States
United States
United States
United States
United States
United States
United States
United States
United States
MATOS NEGRON, TAINA DEL MAR
2014-10-2014519053ANDROGEN RECEPTOR MODULATOR COMPOUNDS AND METHODSLigand Pharmaceuticals IncorporatedPatented Case2016-06-079359285US20150099720A1
Lin Zhi
Robert I. Higuchi
Cornelis Arjan Van Oeveren
Thomas Lot Stevens Lau
United States
United States
United States
United States
CHANDRAKUMAR, NIZAL S
2014-10-0614507693FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USECydex Pharmaceuticals, Inc.Patented Case2015-09-089125945US20150025243A1
Gerold L. Mosher
Rebecca L. Wedel
Karen T. Johnson
Stephen G. Machatha
Jane A. Cowee
Daniel J. Cushing
United States
United States
United States
United States
United States
United States
SHIAO, REI TSANG
2014-09-1714489348SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS AND METHODS OF PREPARATION THEREOFCYDEX PHARMACEUTICALS, INC.Patented Case2017-04-119617352US20150050355A1
James D. Pipkin
Gerold L. Mosher
Douglas B. Hecker
United States
United States
United States
OLSON, ANDREA STEFFEL
2014-09-1214485195PHARMACEUTICAL COMPOSITIONS COMPRISING PRASUGREL AND CYCLODEXTRIN DERIVATIVES AND METHODS OF MAKING AND USING THE SAMECydex Pharmaceuticals, Inc.Patented Case2016-07-269399067US20150005341A1
Gerold L. Mosher
Stephen G. Machatha
Daniel J. Cushing
United States
United States
United States
MAIER, LEIGH C
2014-08-2714381568ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAMECydex Pharmaceuticals Inc.Patented Case2016-11-159493582US20150045311A1
Vincent D. Antle
Alvaro Lopes
Daniel Monteiro
United States
Portugal
Portugal
OLSON, ANDREA STEFFEL
2014-08-1414378953MANUFACTURING PROCESS FOR CYCLODEXTRIN DERIVATIVESCYDEX PHARMACEUTICALS, INC.Patented Case2017-09-059751957US20160009826A1
Vincent D. Antle
Jose R Matos
United States
United States
OLSON, ANDREA STEFFEL
2014-05-0914357551METHODS AND COMPOSITIONS ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTORLigand Pharmaceuticals IncorporatedPatented Case2016-11-159492430US20140296292A1
Lin Zhi
Keith Marschke
Virginia H. Grant
Steven L. Roach
Yixing Shen
Jason C. Pickens
Bijan Pedram
C. Arjan van Oeveren
Lino J. Valdez
Andrew R. Hudson
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
JACKSON, SHAWQUIA
2014-04-2814263237SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2015-09-229139520US20140350065A1
Lin Zhi
United States
MCDOWELL, BRIAN E
2014-03-2814229523Injectable Nitrogen Mustard Compositions Comprising a Cyclodextrin Derivative and Methods of Making and Using the SameCydex Pharmaceuticals, Inc.Patented Case2021-06-0111020363US20140213650A1
James D. Pipkin
Stephen G. Machatha
United States
United States
ARNOLD, ERNST V
2014-01-0314147457NOVEL ANTAGONISTS OF THE GLUCAGON RECEPTORMetabasis Therapeutics, Inc.Patented Case2015-10-279169201US20140135400A1
Jorge E. Gomez-Galeno
Raja K. Reddy
Paul D. van Poelje
Robert Huerta Lemus
Thanh Huu Nguyen
Matthew P. Grote
Qun Dang
Scott J. Hecker
Venkat Reddy Mali
Mingwei Chen
Zhili Sun
Serge Henri Boyer
Haiqing Li
William Craigo
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
OTTON, ALICIA L
2013-12-2014137318HETEROCYCLE AMINES AND USES THEREOFLigand Pharmaceuticals IncorporatedPatented Case2016-02-239266874US20140155379A1
Koc-Kan Ho
David Diller
Jeffrey J. Letourneau
Brian F. McGuinness
Andrew G. Cole
David Rosen
Cornelis A. van Oeveren
Jason C. Pickens
Lin Zhi
Yixing Shen
Bijan Pedram
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
United States
MORRIS, PATRICIA L
2013-12-1614108169INJECTABLE MELPHALAN COMPOSITIONS COMPRISING A CYCLODEXTRIN DERIVATIVE AND METHODS OF MAKING AND USING THE SAMECYDEX PHARMACEUTICALS, INC.Patented Case2021-03-0910940128US20140221488A1
James D. Pipkin
Stephen G. Machatha
United States
United States
ARNOLD, ERNST V
2013-08-2313974937ANDROGEN RECEPTOR MODULATOR COMPOUNDS AND METHODSLigand Pharmaceuticals IncorporatedPatented Case2014-10-218865918US20140005186A1
Lin Zhi
Robert I. Higuchi
Cornelis Arjan Van Oeveren
Thomas Lot Stevens Lau
United States
United States
United States
United States
CHANDRAKUMAR, NIZAL S
2013-03-1113794677SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS AND METHODS OF PREPARATION THEREOFCyDex Pharmaceuticals, Inc.Patented Case2014-09-098829182US20130288054A1
James D. Pipkin
Gerold L. Mosher
Douglas B. Hecker
United States
United States
United States
OLSON, ANDREA STEFFEL
2013-03-1113794652DPI FORMULATION CONTAINING SULFOALKYL ETHER CYCLODEXTRINCYDEX PHARMACEUTICALS, INC.Patented Case2018-11-0610117940US20130197105A1
James D. Pipkin
Gerold L. Mosher
Douglas B. Hecker
United States
United States
United States
KARPINSKI, LUKE E
2013-03-0713789598SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONSCYDEX PHARMACEUTICALS, INC.Patented Case2015-12-019200088US20130184357A1
Vincent D. Antle
United States
OLSON, ANDREA STEFFEL
2012-12-1413715754BIARYL OXYACETIC ACID COMPOUNDSLIGAND PHARMACEUTICALS INC.Patented Case2014-09-028822467US20130102609A1
Brian F. McGuinness
Koc-Kan Ho
Suresh Babu
Guizhen Dong
Jingqi Duo
Thuy X.H. Le
Kurt W. Saionz
United States
United States
United States
United States
United States
United States
United States
SHTERENGARTS, SAMANTHA L
2012-11-3013689898FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USECYDEX PHARMACEUTICALS, INC.Patented Case2014-10-078853236US20130129700A1
Gerold L. MOSHER
Rebecca L. Wedel
Karen T. Johnson
Stephen G. Machatha
Jane A. Cowee
Daniel J. Cushing
United States
United States
United States
United States
United States
United States
SHIAO, REI TSANG
2012-11-1413676744Inhalant Formulation Containing Sulfoalkyl Ether Cyclodextrin and CorticosteroidCyDex Pharmaceuticals, Inc.Patented Case2018-12-2510159752US20130303498A1
James D. PIPKIN
Rupert O. ZIMMERER
Diane O. THOMPSON
Gerold L. MOSHER
United States
United States
United States
United States
KARPINSKI, LUKE E
2012-10-2313694063SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOFLIGAND PHARMACEUTICALS INCORPORATEDPatented Case2014-06-108748633US20130184206A1
Lin Zhi
United States
MCDOWELL, BRIAN E