LIGAND PHARMACEUTICALS INCORPORATED Active Patents
93 granted patents the USPTO still lists as patented, newest filing first, as the USPTO Open Data Portal records them; the company is the first-named applicant. The application number opens the full record at Patent Center.
- 2024-03-05: Application 18595919; Invention USE OF THYROID BETA-AGONISTS; Applicant Metabasis Therapeutics, Inc.; Status Patented Case.
- 2023-06-23: Application 18340177; Invention TOPICAL ANTIVIRAL COMPOSITIONS, DELIVERY SYSTEMS, AND METHODS OF USING THE SAME; Applicant Ligand Pharmaceuticals Incorporated; Status Patented Case.
- 2023-03-22: Application 18246284; Invention ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME; Applicant CYDEX PHARMACEUTICALS, INC.; Status Patented Case.
- 2022-10-19: Application 17996613; Invention BENZYLOXY PHOSPH(ON)ATE COMPOUNDS; Applicant Ligand Pharmaceuticals Incorporated; Status Patented Case.
| Filed | Application | Invention | Applicant | Status | Granted | Patent | Published as | Inventor name | Inventor country | Examiner |
|---|---|---|---|---|---|---|---|---|---|---|
| 2024-03-05 | 18595919 | USE OF THYROID BETA-AGONISTS | Metabasis Therapeutics, Inc. Viking Therapeutics, Inc. | Patented Case | 2025-10-14 | 12440502 | US20250000880A1 | Brian Lian Rochelle Hanley Misha DINERMAN Mark Erion Serge Boyer Hongjian Jiang | United States United States United States United States United States China | RAMACHANDRAN, UMAMAHESWARI |
| 2023-06-23 | 18340177 | TOPICAL ANTIVIRAL COMPOSITIONS, DELIVERY SYSTEMS, AND METHODS OF USING THE SAME | Ligand Pharmaceuticals Incorporated | Patented Case | 2025-09-02 | 12403087 | US20230330008A1 | Kimberly McHale Ryan Doxey Nathan Stasko | United States United States United States | MAEWALL, SNIGDHA |
| 2023-03-22 | 18246284 | ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2026-08-04 | 12698348 | US20230357451A1 | Vincent D. ANTLE Andre FERNANDES Mariana RODRIGUES Claudio VILELA | United States Portugal Portugal Portugal | WARD, PAUL V |
| 2022-10-19 | 17996613 | BENZYLOXY PHOSPH(ON)ATE COMPOUNDS | Ligand Pharmaceuticals Incorporated | Patented Case | 2026-02-17 | 12552820 | US20230159574A1 | Lin Zhi | United States | MCINTOSH III, TRAVISS C |
| 2022-06-08 | 17835828 | NUCLEOTIDE PRODRUG COMPOUNDS | Ligand Pharmaceuticals Incorporated | Patented Case | 2023-01-31 | 11566041 | US20220298198A1 | Lin Zhi | United States | BERRY, LAYLA D |
| 2022-05-11 | 17776199 | ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME | CyDex Pharmaceuticals, Inc. | Patented Case | 2026-07-07 | 12674005 | US20230002513A1 | Vincent D. Antle | United States | CRAIGO, BAHAR ALAWI |
| 2022-05-06 | 17738621 | USE OF THYROID BETA-AGONISTS | Metabasis Therapeutics, Inc. Viking Therapeutics, Inc. | Patented Case | 2024-04-09 | 11951114 | US20220257618A1 | BRIAN LIAN Rochelle Hanley Misha Dinerman Mark Erion Serge Boyer Hongjian Jiang | United States United States United States United States United States China | RAMACHANDRAN, UMAMAHESWARI |
| 2021-10-28 | 17513093 | HETEROCYCLE AMINES AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2023-10-03 | 11773110 | US20220119413A1 | Koc-Kan Ho David Diller Jeffrey J. Letourneau Brian F. McGuinness Andrew G. Cole David Rosen Cornelis A. van Oeveren Jason C. Pickens Lin Zhi Yixing Shen Bijan Pedram | United States United States United States United States United States United States United States United States United States United States United States | KIFLE, BRUCK |
| 2021-10-18 | 17604729 | CRYSTALLINE FORMS AND METHODS OF PRODUCING CRYSTALLINE FORMS OF A COMPOUND | Ligand Pharmaceuticals Incorporated | Patented Case | 2025-06-03 | 12319651 | US20220204448A1 | Lin Zhi Henri Sasmor | United States United States | ISMAIL, REHANA |
| 2021-09-03 | 17465929 | TUNABLE NITRIC OXIDE-RELEASING MACROMOLECULES HAVING MULTIPLE NITRIC OXIDE DONOR STRUCTURES | Ligand Pharmaceuticals Incorporated The University of North Carolina at Chapel Hill | Patented Case | 2025-12-23 | 12503428 | US20210395191A1 | Mark Schoenfisch Yuan Lu Nathan Stasko Jian Bao | United States United States United States United States | XU, JIANGTIAN |
| 2021-07-28 | 17387929 | NASAL AND OPHTHALMIC DELIVERY OF AQUEOUS CORTICOSTEROID SOLUTIONS | CyDex Pharmaceuticals, Inc. | Patented Case | 2025-07-29 | 12370352 | US20220339414A1 | James D. Pipkin Rupert O. Zimmerer JR. John M. Siebert | United States United States United States | WERTZ, ASHLEE ELIZABETH |
| 2021-01-14 | 17148785 | Azetidine Derivatives | Ligand UK Development Limited | Patented Case | 2025-03-11 | 12246014 | US20210267974A1 | Stephen Roughley Steven Walls Terance Hart Rachel Parsons Paul Brough Christopher Graham Alba Macias | United Kingdom United Kingdom United Kingdom United Kingdom United Kingdom United Kingdom United Kingdom | COPPINS, JANET L |
| 2020-11-24 | 17103328 | FRACTIONATED ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME | CyDex Pharmaceuticals, Inc. | Patented Case | 2023-10-24 | 11795241 | US20210147582A1 | Vincent D. Antle Charles Alan Watson David W. Miles | United States United States United States | MAIER, LEIGH C |
| 2020-10-15 | 17071273 | IMIDAZO-FUSED HETEROCYCLES AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2024-01-02 | 11858938 | US20210040102A1 | Lin Zhi | United States | KANTAMNENI, SHOBHA |
| 2020-09-15 | 17021909 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS | CyDex Pharmaceuticals, Inc. | Patented Case | 2023-11-07 | 11806402 | US20210093727A1 | Vincent D. Antle | United States | OLSON, ANDREA STEFFEL |
| 2020-08-12 | 16969521 | GLUCAGON RECEPTOR ANTAGONISTS | LIGAND PHARMACEUTICALS INCORPORATED | Patented Case | 2025-01-28 | 12208071 | US20210121422A1 | Lin Zhi Ian Henderson Joseph Kaloko Martin Osterhout | United States United States United States United States | COFFA, SERGIO |
| 2020-08-03 | 16983617 | SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2022-06-14 | 11358931 | US20200361866A1 | Lin Zhi | United States | MCDOWELL, BRIAN E |
| 2020-07-10 | 16925926 | METHODS AND COMPOSITIONS ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR | Ligand Pharmaceuticals, Inc. | Patented Case | 2022-08-16 | 11413274 | US20210046045A1 | Lin Zhi Keith Marschke Virginia H. Grant Steven L. Roach Yixing Shen Jason C. Pickens Bijan Pedram Cornelis Arjan van Oeveren Lino J. Valdez Andrew R. Hudson | United States United States United States United States United States United States United States United States United States United States | JACKSON, SHAWQUIA |
| 2020-07-08 | 16960681 | ACETAL COMPOUNDS AND THERAPEUTIC USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2024-04-30 | 11970482 | US20200339551A1 | Lin Zhi | United States | SEAMAN, D MARGARET M |
| 2020-05-15 | 16875855 | DPI FORMULATION CONTAINING SULFOALKYL ETHER CYCLODEXTRIN | CyDex Pharmaceuticals, Inc. | Patented Case | 2022-10-11 | 11464862 | US20200276314A1 | James D. Pipkin Gerold L. Mosher Douglas B. Hecker | United States United States United States | HIRT, ERIN E |
| 2020-01-24 | 16752400 | MANUFACTURING PROCESS FOR CYCLODEXTRIN DERIVATIVES | CyDex Pharmaceuticals, Inc. | Patented Case | 2021-12-28 | 11208500 | US20200157252A1 | Vincent D. Antle Jose R. Matos | United States United States | OLSON, ANDREA STEFFEL |
| 2020-01-07 | 16735988 | HETEROCYCLE AMINES AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2021-11-30 | 11186593 | US20200216468A1 | Koc-Kan Ho David Diller Jeffrey J. Letourneau Brian F. McGuinness Andrew G. Cole David Rosen Cornelis A. van Oeveren Jason C. Pickens Lin Zhi Yixing Shen Bijan Pedram | United States United States United States United States United States United States United States United States United States United States United States | KIFLE, BRUCK |
| 2019-12-27 | 16728840 | Injectable Nitrogen Mustard Compositions Comprising a Cyclodextrin Derivative and Methods of Making and Using the Same | Cydex Pharmaceuticals, Inc. | Patented Case | 2020-12-15 | 10864183 | US20200268698A1 | James D. Pipkin Stephen G. Machatha | United States United States | ARNOLD, ERNST V |
| 2019-11-01 | 16672170 | COMPOSITION CONTAINING SULFOALKYL ETHER CYCLODEXTRIN AND LATANOPROST | CyDex Pharmaceuticals, Inc. | Patented Case | 2022-09-06 | 11433082 | US20200179400A1 | Naomi Esaki James D. Pipkin | United States United States | BABSON, NICOLE PLOURDE |
| 2019-09-16 | 16572493 | METHODS AND COMPOSITIONS FOR MODULATING HORMONE LEVELS | Ligand Pharmaceuticals Incorporated | Patented Case | 2020-12-29 | 10874638 | US20200009112A1 | Lin Zhi | United States | WEDDINGTON, KEVIN E |
| 2019-08-30 | 16557768 | PRODRUG COMPOUNDS AND THEIR USES | LIGAND PHARMACEUTICALS INCORPORATED | Patented Case | 2022-03-22 | 11278559 | US20190388452A1 | Lin Zhi | United States | LEWIS, PATRICK T |
| 2019-03-14 | 16333576 | FORMULATIONS CONTAINING ACETAMINOPHEN AND SULFOALKYL ETHER CYCLODEXTRIN | CyDex Pharmaceuticals, Inc. | Patented Case | 2026-01-20 | 12527755 | US20190255000A1 | James D. Pipkin Gerold L. Mosher Roger A. Rajewski | United States United States United States | CHONG, YONG SOO |
| 2019-02-28 | 16289241 | GLUCAGON ANTAGONISTS | Metabasis Therapeutics, Inc. | Patented Case | 2022-06-07 | 11352321 | US20190330144A1 | Jorge E GOMEZ-GALENO Scott J. HECKER Qun DANG Mali Venkat REDDY Zhili SUN Matthew P. GROTE Thanh Huu NGUYEN Robert Huerta LEMUS Haiqing LI | United States United States United States United States United States United States United States United States United States | JAVANMARD, SAHAR |
| 2019-02-08 | 16271735 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS AND METHODS OF PREPARATION THEREOF | CyDex Pharmaceuticals, Inc. | Patented Case | 2020-07-07 | 10703826 | US20190169316A1 | James D. Pipkin Gerold L. Mosher Douglas B. Hecker | United States United States United States | OLSON, ANDREA STEFFEL |
| 2018-12-05 | 16210561 | INHALANT FORMULATION CONTAINING SULFOALKYL ETHER CYCLODEXTRIN AND CORTICOSTEROID | CyDex Pharmaceuticals, Inc. | Patented Case | 2020-10-13 | 10799599 | US20190105404A1 | James D. PIPKIN Rupert O. ZIMMERER Diane O. THOMPSON Gerold L. MOSHER | United States United States United States United States | HAGHIGHATIAN, MINA |
| 2018-11-19 | 16195782 | THYROMIMETICS FOR THE TREATMENT OF FATTY LIVER DISEASES | Metabasis Therapeutics, Inc. | Patented Case | 2021-02-23 | 10925885 | US20190083515A1 | Edward E. Cable Mark D. Erion | United States United States | KATAKAM, SUDHAKAR |
| 2018-11-05 | 16181233 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS | CyDex Pharmaceuticals, Inc. | Patented Case | 2020-09-22 | 10780177 | US20190070303A1 | Vincent D. Antle | United States | OLSON, ANDREA STEFFEL |
| 2018-10-19 | 16095228 | USE OF THYROID BETA-AGONISTS | Metabasis Therapeutics, Inc. Viking Therapeutics, Inc. | Patented Case | 2022-06-07 | 11351183 | US20190321379A1 | Brian Lian Rochelle Hanley Misha Dinerman Mark Erion Serge Boyer Hongjian Jiang | United States United States United States United States United States China | RAMACHANDRAN, UMAMAHESWARI |
| 2018-10-01 | 16148798 | SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2020-08-04 | 10730831 | US20190040006A1 | Lin Zhi | United States | MCDOWELL, BRIAN E |
| 2018-09-10 | 16126199 | METHODS AND COMPOSITIONS ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR | Ligand Pharmaceuticals, Inc. | Patented Case | 2020-08-11 | 10736875 | US20180369197A1 | Lin Zhi Keith Marschke Virginia H. Grant Steven L. Roach Yixing Shen Jason C. Pickens Bijan Pedram Cornelis Arjan van Oeveren Lino J. Valdez Andrew R. Hudson | United States United States United States United States United States United States United States United States United States United States | JACKSON, SHAWQUIA |
| 2018-08-08 | 16058778 | THYROID HORMONE RECEPTOR AGONIST AND USE THEREOF | Metabasis Therapeutics, Inc. | Patented Case | 2019-09-24 | 10420781 | US20180344752A1 | Mark Erion Hongjian Jiang Serge Henri Boyer | United States China United States | SHTERENGARTS, SAMANTHA L |
| 2018-08-02 | 16053550 | ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME | CyDex Pharmaceuticals, Inc. | Patented Case | 2020-10-13 | 10800861 | US20180346609A1 | Vincent D. Antle Álvaro Lopes Daniel Monteiro | United States Portugal Portugal | OLSON, ANDREA STEFFEL |
| 2018-07-24 | 16043833 | FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USE | Cydex Pharmaceuticals, Inc. | Patented Case | 2019-12-24 | 10512697 | US20180326090A1 | Gerold L. Mosher Rebecca L. Wedel Karen T. Johnson Stephen G. Machatha Jane A. Cowee Daniel J. Cushing | United States United States United States United States United States United States | SHIAO, REI TSANG |
| 2018-07-02 | 16025199 | INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE 1 (DGAT-1) AND USES THEREOF | Metabasis Therapeutics, Inc. | Patented Case | 2020-07-14 | 10709718 | US20180303856A1 | K. Raja Reddy Jeff Stebbins Serge H. Boyer Mark D. Erion Scott J. Hecker Nicholas Brian Raffaele Brett C. Bookser Venkat Reddy Mali | United States United States United States United States United States United States United States United States | MURRAY, JEFFREY H |
| 2018-06-22 | 16015925 | HETEROCYCLE AMINES AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2020-03-31 | 10604533 | US20180298031A1 | Koc-Kan Ho David Diller Jeffrey J. Letourneau Brian F. McGuinness Andrew G. Cole David Rosen Cornelis A. van Oeveren Jason C. Pickens Lin Zhi Yixing Shen Bijan Pedram | United States United States United States United States United States United States United States United States United States United States United States | KIFLE, BRUCK |
| 2018-06-11 | 16005601 | PRODRUG COMPOUNDS AND USES THEROF | Ligand Pharmaceuticals Inc. | Patented Case | 2018-12-11 | 10150788 | US20180291050A1 | Lin Zhi | United States | ROZOF, TIMOTHY R |
| 2018-02-28 | 15908504 | METHODS OF TREATMENT ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR | LIGAND PHARMACEUTICALS INCORPORATED | Patented Case | 2019-09-24 | 10420748 | US20180185333A1 | Keith B. Marschke Lin Zhi | United States United States | WEDDINGTON, KEVIN E |
| 2017-11-17 | 15817056 | INHALANT FORMULATION CONTAINING SULFOALKYL ETHER CYCLODEXTRIN AND CORTICOSTEROID | CyDex Pharmaceuticals, Inc. | Patented Case | 2019-02-19 | 10207008 | US20180154015A1 | James D. Pipkin Rupert O. Zimmerer Diane O. Thompson Gerold L. Mosher | United States United States United States United States | SCHLIENTZ, NATHAN W |
| 2017-09-29 | 15721556 | GLUCAGON ANTAGONISTS | Metabasis Therapeutics, Inc. | Patented Case | 2019-03-05 | 10221130 | US20180022695A1 | Jorge E. Gomez-Galeno Scott J. Hecker Qun Dang Mali Venkat Reddy Zhili Sun Matthew P. Grote Thanh Huu Nguyen Robert Huerta Lemus Haiqing Li | United States United States United States United States United States United States United States United States United States | MATOS NEGRON, TAINA DEL MAR |
| 2017-08-31 | 15693248 | MANUFACTURING PROCESS FOR CYCLODEXTRIN DERIVATIVES | CyDex Pharmaceuticals, Inc. | Patented Case | 2020-04-28 | 10633462 | US20180051098A1 | Vincent D. Antle Jose R. Matos | United States United States | OLSON, ANDREA STEFFEL |
| 2017-08-25 | 15687407 | METHOD FOR TREATING DISORDERS ASSOCIATED WITH GLOMERULAR FUNCTION | Ligand Pharmaceuticals Inc. | Patented Case | 2018-06-12 | 9993461 | US20170354646A1 | Jinkun Zhang Zofia E. Dziewanowska Rene Belder Ian Henderson Joseph B. Bogardus Zhaoying Zhang | United States United States United States United States United States United States | HARTSFIELD, KATHRIEN ANN |
| 2017-05-09 | 15590884 | SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2018-10-23 | 10106500 | US20170247325A1 | Lin Zhi | United States | MCDOWELL, BRIAN E |
| 2017-05-09 | 15590813 | DERIVATIVES OF URIDINE 5'-CYCLOPHOSPHATE USEFUL TO TREAT HEPATITIS C VIRAL INFECTIONS | Ligand Pharmaceuticals Incorporated | Patented Case | 2018-06-19 | 10000522 | US20170334942A1 | Lin Zhi | United States | MCINTOSH III, TRAVISS C |
| 2017-03-09 | 15454967 | FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USE | Cydex Pharmaceuticals, Inc. | Patented Case | 2018-07-31 | 10034947 | US20170173178A1 | Gerold L. Mosher Rebecca L. Wedel Karen T. Johnson Stephen G. Machatha Jane A. Cowee Daniel J. Cushing | United States United States United States United States United States United States | SHIAO, REI TSANG |
| 2017-03-02 | 15448411 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS AND METHODS OF PREPARATION THEREOF | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2019-02-12 | 10202468 | US20170172926A1 | James D. Pipkin Gerold L. Mosher Douglas B. Hecker | United States United States United States | OLSON, ANDREA STEFFEL |
| 2017-02-21 | 15505428 | FRACTIONATED ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME | CyDex Pharmaceuticals, Inc. | Patented Case | 2020-12-01 | 10851184 | US20170275388A1 | Vincent D. Antle Charles Alan Watson David W. Miles | United States United States United States | MAIER, LEIGH C |
| 2016-12-29 | 15323080 | PRODRUG COMPOUNDS AND USES THEROF | LIGAND PHARMACEUTICALS, INC. | Patented Case | 2018-06-12 | 9994600 | US20170158725A1 | Lin Zhi | United States | ROZOF, TIMOTHY R |
| 2016-11-14 | 15351272 | ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME | Cydex Pharmaceuticals, Inc. | Patented Case | 2019-06-18 | 10323103 | US20170158781A1 | Vincent D. Antle Alvaro Lopes Daniel Monteiro | United States Portugal Portugal | OLSON, ANDREA STEFFEL |
| 2016-08-25 | 15247164 | METHODS AND COMPOSITIONS ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR | Ligand Pharmaceuticals, Inc. | Patented Case | 2018-10-30 | 10111859 | US20160374989A1 | Lin Zhi Keith Marschke Virginia H. Grant Steven L. Roach Yixing Shen Jason C. Pickens Bijan Pedram Cornelius Arjan van Oeveren Lino J. Valdez Andrew R. Hudson | United States United States United States United States United States United States United States United States United States United States | JACKSON, SHAWQUIA |
| 2016-08-12 | 15118821 | PRODRUG COMPOUNDS AND THEIR USES | LIGAND PHARMACEUTICALS, INC. | Patented Case | 2019-10-22 | 10449210 | US20170056429A1 | Lin Zhi | United States | LEWIS, PATRICK T |
| 2016-08-10 | 15233748 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS | CyDex Pharmaceuticals, Inc. | Patented Case | 2017-09-05 | 9750822 | US20160346405A1 | Vincent D. Antle | United States | MAIER, LEIGH C |
| 2016-07-14 | 15111741 | METHODS AND COMPOSITIONS FOR MODULATING HORMONE LEVELS | LIGAND PHARMACEUTICALS INCORPORATED | Patented Case | 2019-10-15 | 10441567 | US20160338995A1 | Lin Zhi | United States | WEDDINGTON, KEVIN E |
| 2016-06-13 | 15181190 | PHARMACEUTICAL COMPOSITIONS COMPRISING PRASUGREL AND CYCLODEXTRIN DERIVATIVES AND METHODS OF MAKING AND USING THE SAME | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2018-10-30 | 10111863 | US20170007586A1 | Gerold L. Mosher Stephen G. Machatha Daniel J. Cushing | United States United States United States | MAIER, LEIGH C |
| 2016-05-11 | 15151740 | INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE 1 (DGAT-1) AND USES THEREOF | METABASIS THERAPEUTICS, INC. | Patented Case | 2018-07-31 | 10034891 | US20160263132A1 | K. RAJA REDDY JEFF STEBBINS SERGE H. BOYER MARK D. ERION SCOTT J. HECKER NICHOLAS BRIAN RAFFAELE BRETT C. BOOKSER VENKAT REDDY MALI | United States United States United States United States United States United States United States United States | MURRAY, JEFFREY H |
| 2016-05-05 | 15034757 | DERIVATIVES OF URIDINE 5'-CYCLOPHOSPHATE USEFUL TO TREAT HEPATITIS C VIRAL INFECTIONS | LIGAND PHARMACEUTICALS INCORPORATED | Patented Case | 2017-06-13 | 9676809 | US20160347783A1 | Lin Zhi | United States | MCINTOSH III, TRAVISS C |
| 2016-03-15 | 15070718 | IMIDAZO-FUSED HETEROCYCLES AND USES THEREOF | Ligand Pharmaceuticals, Inc. | Patented Case | 2020-10-20 | 10807983 | US20160297824A1 | Lin Zhi | United States | KANTAMNENI, SHOBHA |
| 2016-01-26 | 15006940 | HETEROCYCLE AMINES AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2018-07-24 | 10030034 | US20160347767A1 | Koc-Kan Ho David Diller Jeffrey J. Letourneau Brian F. McGuinness Andrew G. Cole David Rosen Cornelis A. van Oeveren Jason C. Pickens Lin Zhi Yixing Shen Bijan Pedram | United States United States United States United States United States United States United States United States United States United States United States | KIFLE, BRUCK |
| 2015-11-30 | 14954772 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS | CyDex Pharmaceuticals, Inc. | Patented Case | 2018-11-06 | 10117951 | US20160158384A1 | Vincent D. Antle | United States | OLSON, ANDREA STEFFEL |
| 2015-09-11 | 14775587 | METHODS OF TREATMENT ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR | LIGAND PHARMACEUTICALS INCORPORATED | Patented Case | 2018-05-08 | 9962370 | US20160022638A1 | Keith B. Marschke Lin Zhi | United States United States | WEDDINGTON, KEVIN E |
| 2015-09-04 | 14846049 | FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USE | Cydex Pharmaceuticals, Inc. | Patented Case | 2017-04-18 | 9623045 | US20160058786A1 | Gerold L. Mosher Rebecca L. Wedel Karen T. Johnson Stephen G. Machatha Jane A. Cowee Daniel J. Cushing | United States United States United States United States United States United States | SHIAO, REI TSANG |
| 2015-08-14 | 14827228 | SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2017-06-13 | 9675583 | US20160038461A1 | Lin Zhi | United States | MCDOWELL, BRIAN E |
| 2015-05-15 | 14713930 | HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES | LIGAND PHARMACEUTICALS INC. | Patented Case | 2017-04-18 | 9622991 | US20150252043A1 | Lin Zhi Andrew R. Hudson Cornelis A. Van Oeveren Steven L. Roach Bijan Pedram Yixing Shen Lino J. Valdez Jillian Basinger Virginia Heather Sharron Grant Jason C. Pickens | United States United States United States United States United States United States United States United States United States United States | SHTERENGARTS, SAMANTHA L |
| 2015-04-21 | 14437439 | ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2018-08-07 | 10040872 | US20150284479A1 | Vincent D. Antle Álvaro Lopes Daniel Monteiro | United States Portugal Portugal | OLSON, ANDREA STEFFEL |
| 2015-03-13 | 14428151 | NOVEL NUCLEOTIDE PRODRUG COMPOUNDS AND USE | LIGAND PHARMACEUTICALS INC. | Patented Case | 2016-05-03 | 9326991 | US20150246068A1 | Lin Zhi K. Raja Reddy | United States United States | MCINTOSH III, TRAVISS C |
| 2015-02-25 | 14631768 | METHOD FOR TREATING GLOMERULOSCLEROSIS | Ligand Pharmaceuticals Inc. | Patented Case | 2017-05-30 | 9662312 | US20150164865A1 | Jinkun Zhang Zofia E. Dziewanowska Rene Belder Ian Henderson Joseph B. Bogardus Zhaoying Zhang | United States United States United States United States United States United States | HARTSFIELD, KATHRIEN ANN |
| 2015-02-23 | 14628373 | INHIBITORS OF DIACYLGLYCEROL O-ACYLTRANSFERASE 1 (DGAT-1) AND USES THEREOF | METABASIS THERAPEUTICS, INC. | Patented Case | 2016-05-17 | 9340566 | US20150166590A1 | K. RAJA REDDY JEFF STEBBINS SERGE H. BOYER MARK D. ERION SCOTT J. HECKER NICHOLAS BRIAN RAFFAELE BRETT C. BOOKSER VENKAT REDDY MALI | United States United States United States United States United States United States United States United States | MURRAY, JEFFREY H |
| 2014-12-29 | 14585073 | NOVEL ACTIVATORS OF GLUCOKINASE | Metabasis Therapeutics, Inc. | Patented Case | 2016-12-20 | 9522926 | US20150119365A1 | Feng Tian Qun Dang G. Sridhar Prasad Wenyu Li Brett C. Bookser Nicholas Brian Raffaele Mark D. Erion | United States United States United States United States United States United States United States | BALASUBRAMANIAN, VENKATARAMAN |
| 2014-11-26 | 14555503 | GLUCAGON ANTAGONISTS | Metabasis Therapeutics, Inc. | Patented Case | 2017-10-10 | 9783494 | US20150087680A1 | Jorge E. Gomez-Galeno Scott J. Hecker Qun Dang Mali Venkat Reddy Zhili Sun Matthew P. Grote Thanh Huu Nguyen Robert Huerta Lemus Haiqing Li | United States United States United States United States United States United States United States United States United States | MATOS NEGRON, TAINA DEL MAR |
| 2014-10-20 | 14519053 | ANDROGEN RECEPTOR MODULATOR COMPOUNDS AND METHODS | Ligand Pharmaceuticals Incorporated | Patented Case | 2016-06-07 | 9359285 | US20150099720A1 | Lin Zhi Robert I. Higuchi Cornelis Arjan Van Oeveren Thomas Lot Stevens Lau | United States United States United States United States | CHANDRAKUMAR, NIZAL S |
| 2014-10-06 | 14507693 | FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USE | Cydex Pharmaceuticals, Inc. | Patented Case | 2015-09-08 | 9125945 | US20150025243A1 | Gerold L. Mosher Rebecca L. Wedel Karen T. Johnson Stephen G. Machatha Jane A. Cowee Daniel J. Cushing | United States United States United States United States United States United States | SHIAO, REI TSANG |
| 2014-09-17 | 14489348 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS AND METHODS OF PREPARATION THEREOF | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2017-04-11 | 9617352 | US20150050355A1 | James D. Pipkin Gerold L. Mosher Douglas B. Hecker | United States United States United States | OLSON, ANDREA STEFFEL |
| 2014-09-12 | 14485195 | PHARMACEUTICAL COMPOSITIONS COMPRISING PRASUGREL AND CYCLODEXTRIN DERIVATIVES AND METHODS OF MAKING AND USING THE SAME | Cydex Pharmaceuticals, Inc. | Patented Case | 2016-07-26 | 9399067 | US20150005341A1 | Gerold L. Mosher Stephen G. Machatha Daniel J. Cushing | United States United States United States | MAIER, LEIGH C |
| 2014-08-27 | 14381568 | ALKYLATED CYCLODEXTRIN COMPOSITIONS AND PROCESSES FOR PREPARING AND USING THE SAME | Cydex Pharmaceuticals Inc. | Patented Case | 2016-11-15 | 9493582 | US20150045311A1 | Vincent D. Antle Alvaro Lopes Daniel Monteiro | United States Portugal Portugal | OLSON, ANDREA STEFFEL |
| 2014-08-14 | 14378953 | MANUFACTURING PROCESS FOR CYCLODEXTRIN DERIVATIVES | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2017-09-05 | 9751957 | US20160009826A1 | Vincent D. Antle Jose R Matos | United States United States | OLSON, ANDREA STEFFEL |
| 2014-05-09 | 14357551 | METHODS AND COMPOSITIONS ASSOCIATED WITH THE GRANULOCYTE COLONY-STIMULATING FACTOR RECEPTOR | Ligand Pharmaceuticals Incorporated | Patented Case | 2016-11-15 | 9492430 | US20140296292A1 | Lin Zhi Keith Marschke Virginia H. Grant Steven L. Roach Yixing Shen Jason C. Pickens Bijan Pedram C. Arjan van Oeveren Lino J. Valdez Andrew R. Hudson | United States United States United States United States United States United States United States United States United States United States | JACKSON, SHAWQUIA |
| 2014-04-28 | 14263237 | SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2015-09-22 | 9139520 | US20140350065A1 | Lin Zhi | United States | MCDOWELL, BRIAN E |
| 2014-03-28 | 14229523 | Injectable Nitrogen Mustard Compositions Comprising a Cyclodextrin Derivative and Methods of Making and Using the Same | Cydex Pharmaceuticals, Inc. | Patented Case | 2021-06-01 | 11020363 | US20140213650A1 | James D. Pipkin Stephen G. Machatha | United States United States | ARNOLD, ERNST V |
| 2014-01-03 | 14147457 | NOVEL ANTAGONISTS OF THE GLUCAGON RECEPTOR | Metabasis Therapeutics, Inc. | Patented Case | 2015-10-27 | 9169201 | US20140135400A1 | Jorge E. Gomez-Galeno Raja K. Reddy Paul D. van Poelje Robert Huerta Lemus Thanh Huu Nguyen Matthew P. Grote Qun Dang Scott J. Hecker Venkat Reddy Mali Mingwei Chen Zhili Sun Serge Henri Boyer Haiqing Li William Craigo | United States United States United States United States United States United States United States United States United States United States United States United States United States United States | OTTON, ALICIA L |
| 2013-12-20 | 14137318 | HETEROCYCLE AMINES AND USES THEREOF | Ligand Pharmaceuticals Incorporated | Patented Case | 2016-02-23 | 9266874 | US20140155379A1 | Koc-Kan Ho David Diller Jeffrey J. Letourneau Brian F. McGuinness Andrew G. Cole David Rosen Cornelis A. van Oeveren Jason C. Pickens Lin Zhi Yixing Shen Bijan Pedram | United States United States United States United States United States United States United States United States United States United States United States | MORRIS, PATRICIA L |
| 2013-12-16 | 14108169 | INJECTABLE MELPHALAN COMPOSITIONS COMPRISING A CYCLODEXTRIN DERIVATIVE AND METHODS OF MAKING AND USING THE SAME | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2021-03-09 | 10940128 | US20140221488A1 | James D. Pipkin Stephen G. Machatha | United States United States | ARNOLD, ERNST V |
| 2013-08-23 | 13974937 | ANDROGEN RECEPTOR MODULATOR COMPOUNDS AND METHODS | Ligand Pharmaceuticals Incorporated | Patented Case | 2014-10-21 | 8865918 | US20140005186A1 | Lin Zhi Robert I. Higuchi Cornelis Arjan Van Oeveren Thomas Lot Stevens Lau | United States United States United States United States | CHANDRAKUMAR, NIZAL S |
| 2013-03-11 | 13794677 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS AND METHODS OF PREPARATION THEREOF | CyDex Pharmaceuticals, Inc. | Patented Case | 2014-09-09 | 8829182 | US20130288054A1 | James D. Pipkin Gerold L. Mosher Douglas B. Hecker | United States United States United States | OLSON, ANDREA STEFFEL |
| 2013-03-11 | 13794652 | DPI FORMULATION CONTAINING SULFOALKYL ETHER CYCLODEXTRIN | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2018-11-06 | 10117940 | US20130197105A1 | James D. Pipkin Gerold L. Mosher Douglas B. Hecker | United States United States United States | KARPINSKI, LUKE E |
| 2013-03-07 | 13789598 | SULFOALKYL ETHER CYCLODEXTRIN COMPOSITIONS | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2015-12-01 | 9200088 | US20130184357A1 | Vincent D. Antle | United States | OLSON, ANDREA STEFFEL |
| 2012-12-14 | 13715754 | BIARYL OXYACETIC ACID COMPOUNDS | LIGAND PHARMACEUTICALS INC. | Patented Case | 2014-09-02 | 8822467 | US20130102609A1 | Brian F. McGuinness Koc-Kan Ho Suresh Babu Guizhen Dong Jingqi Duo Thuy X.H. Le Kurt W. Saionz | United States United States United States United States United States United States United States | SHTERENGARTS, SAMANTHA L |
| 2012-11-30 | 13689898 | FORMULATIONS CONTAINING CLOPIDOGREL AND SULFOALKYL ETHER CYCLODEXTRIN AND METHODS OF USE | CYDEX PHARMACEUTICALS, INC. | Patented Case | 2014-10-07 | 8853236 | US20130129700A1 | Gerold L. MOSHER Rebecca L. Wedel Karen T. Johnson Stephen G. Machatha Jane A. Cowee Daniel J. Cushing | United States United States United States United States United States United States | SHIAO, REI TSANG |
| 2012-11-14 | 13676744 | Inhalant Formulation Containing Sulfoalkyl Ether Cyclodextrin and Corticosteroid | CyDex Pharmaceuticals, Inc. | Patented Case | 2018-12-25 | 10159752 | US20130303498A1 | James D. PIPKIN Rupert O. ZIMMERER Diane O. THOMPSON Gerold L. MOSHER | United States United States United States United States | KARPINSKI, LUKE E |
| 2012-10-23 | 13694063 | SELECTIVE ANDROGEN RECEPTOR MODULATORS (SARMS) AND USES THEREOF | LIGAND PHARMACEUTICALS INCORPORATED | Patented Case | 2014-06-10 | 8748633 | US20130184206A1 | Lin Zhi | United States | MCDOWELL, BRIAN E |